平安! 发表于 2011-11-9 19:57
+ U; W. M2 A+ |+ a$ E4 d7 B2 @% UPazopanib (100 mg/kg/day free base equivalent) ( l9 D& w; t$ a
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
) j P5 _& z" w6 D搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。
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" @5 t. c) g! E--------------------- DOSAGE AND ADMINISTRATION ----------------$ C/ Z# ~8 o6 y) }& x& N, d
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
( J& R+ U$ |7 t. r* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
6 e, ~: e, K8 R R: c% [- ?---------------------DOSAGE FORMS AND STRENGTHS --------------
; k3 Q2 Q% H9 c! P! q6 Y* o200 mg tablets. (3) 5 W, Z. q2 \+ X" l
-------------------------------CONTRAINDICATIONS------------------------ |